Local anaesthetic for dentistry

Articaine (أرتيكايين)

Articaine is a local anaesthetic injected by a dentist to prevent pain during dental procedures. Many products also contain adrenaline to prolong numbness and reduce bleeding.

This medicine is used under close medical supervision, usually by a specialist. Never start, stop or change it without your doctor.

What it is used for

  • Local anaesthesia before fillings, extractions or other dental procedures
  • Nerve block or injection around a tooth during dental treatment

How it is used

  • It is given only by a dentist after reviewing your health and medicines
  • Avoid chewing and hot drinks until numbness has worn off so you do not bite your tongue or lip or burn your mouth
  • Follow the dentist's aftercare advice and contact them if numbness persists or unusual symptoms develop

Possible side effects

  • Pain or mild swelling at the injection site and headache
  • Temporary numbness of the lip, tongue or cheek
  • Palpitations, tremor or dizziness from the adrenaline in some products
  • Rarely, seizures, abnormal heart rhythm, severe allergy or blue-grey skin discolouration

Who should not use it

  • Allergy to articaine or a similar local anaesthetic
  • Sulfite allergy when a product containing adrenaline is used

Before and while using it

  • Tell your dentist if you have heart disease, an abnormal rhythm or uncontrolled blood pressure
  • Tell them if you have liver or kidney disease, or a blood disorder such as methaemoglobinaemia or G6PD deficiency
  • Tell the team immediately about ringing in the ears, a metallic taste, numbness around the mouth, confusion or breathing difficulty
  • Get urgent help if the skin or lips turn grey or blue, or facial swelling develops

Medicine interactions

  • Some antidepressants, beta blockers and monoamine oxidase inhibitors can increase adrenaline effects on the heart and blood pressure
  • Other local anaesthetics and some heart rhythm medicines can increase toxicity
  • Medicines that can cause methaemoglobinaemia, such as nitrates, dapsone and some antibiotics, increase the risk

Pregnancy and breastfeeding

  • Tell your dentist if you are pregnant or breastfeeding; they will choose the most suitable product and the lowest suitable amount for the procedure

How to store it

  • The dentist stores and prepares this medicine in the clinic

Get medical help straight away if

  • Your face, lips or tongue swell, or you find it hard to breathe.
  • You get a severe rash, blistering or peeling skin.
  • A side effect worries you or doesn’t go away: contact your doctor or pharmacist.

Questions about this medicine?

Talk to a doctor by video, or send your question by text.

Source: Standard international medicine references

This guide is general information and doesn’t replace advice from your doctor or pharmacist. Don’t start, stop or change a medicine without asking them, and always read the leaflet in the pack.